Uburyo busanzwe bwo kurinda amino

1. Cbz
Benzyloxycarbonyl (Cbz) Irinze Amino
Deprotection ya N-benzyloxycarbonyl (Cbz)
Bikunze gukoreshwa reagent - CbzCl

2. Kugabana
Allyloxycarbonyl (Alloc) yarinze itsinda rya amino

3. Trifluoroacetyl
Trifluoroacetyl yarinze amatsinda ya amino

4. Benzyls
p-mikorerexybenzyl (PMB) irinze amatsinda ya amino
2,4-dimethoxybenzyl irinzwe amatsinda ya amino
Benzyl yarinze amino
Deprotection ya benzyl irinzwe nitsinda rya amino
N-Bn debenzylation kuburyo bwa chloroformate

5. Pht (phthaloyl)
Phthaloyl (Pht) yarinze amatsinda ya amino
Deprotection ya phthaloyl-irinzwe nitsinda rya amino

6. Benzenesulfonyl
Nitrobenzenesulfonyl yarinze amatsinda ya amino
p-toluenesulfonyl (Tos) kurinda amino

7. Trt
Trityl yarinze amino
Deprotection ya trityl ikingiwe nitsinda rya amino

8. Boc
Tert-butoxycarbonyl irinzwe amino itsinda
Deprotection ya N-tert-butoxycarbonyl
Oxalyl Chloride De-Boc

9. Fmoc
Reba mikorerexycarbonyl irinzwe amino itsinda
Bikunze gukoreshwa reagent - Fmoc-Cl

10. SEM
SEM yarinze amino

11. Abandi
Acetamide yarinze amatsinda ya amino
Clauson-Kaas pyrrole synthesis reaction (iyi reaction irashobora gukoreshwa nkuburyo bwo kurinda amatsinda amine, irashobora gusimbuza Boc kurinda kabiri, kandi irahagaze neza)
Bikunze gukoreshwa reagent - benzyl (chloromethyl) ether
Bikunze gukoreshwa reagent - (chloromethyl) methyl ether [MOMCl]
Kurinda Carbamate